Catalog No. :	CL2754
Product Name :	BIX-01294
CAS No. :	935693-62-2
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Chemical Name :
Molecular Formula :	C28H38N6O2
Molecular Weight :	490.64
Molecular Structure :
Appearance :	White to off-white powder
Specification :	98+%
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BIX-01294 is a reversible and highly selective G9a and GLP Histone Methyltransferase inhibitor, with IC₅₀s of of 1.7 μM and 0.9 μM, respectively. BIX-01294 inhibits G9a/GLP by competing for binding with the amino acids N-terminal of the substrate lysine residue. BIX-01294, a (1H-1,4-diazepin-1-yl)-quinazolin-4-yl amine derivative, induces necroptosis and autophagy. BIX-01294 has antitumor activity in recurrent tumor cells。

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